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5⿼ƤʼصٴӦá

ƤʼؿƸݿˣ𰸾Ϊ֤ʴѡA 6⿼Ƥʼصҩ໥á

(1)ͱסӢơƽƽȸҩøյɼӿƤʼشл(2) ܹͪCYP3A ԣӶ߼ѪŨȣ IJεҲӰ죬Ҫ߾衣(3)Ƥʼù B þܴٽżء(4)Ƥʼˮ(簢˾ƥ)ø(5) ʲĴлܼӿڷҩĪ˾Ĵл(6) ùءηͪضCYP3A ƼҪעټ ļʴѡE

8⿼ƤʼصٴӦá

D ΪѡƤʼس˾дͳ֢߷Ӧ⣬мٷ

ϸͷTNF áƤʼΪ˸ҩǿڷν ϷӦҪԭ򡣵ΪҩǷν˵ҪҩųD ƤʼĿǰ֧ΪЧҩҪڰϸܹ֢ Чؿ֧֢״о֣ʹƤʼؿIL-4 IL-5IL-4 ܽṹйأʹƤʼصĻ߳ҩ죬ܵ¼Ե֧ ͺ֢ĸ֧˵ʹڸƤʼҲԽ ĺ߷Ӧԣٴϳ˵ɡ⣬õDZɵ ʴѡC

10⿼ƤʼƵûơ ҩƤʼؿӰ߷ӦĶڣƾϸɹܣ ״Ƥϵͳϸãʹܰϸܽ⣬ܰͽᡢƢܰϸ ĽߡöT ϸԣиT ϸٸɽԿˮ ƽϿ׼ãɻӦԼ֢״Կ ֲ췴ӦʴѡA

12⿼ƼҩӦ֤ ƶƱƽࡣʴѡB 13⿼Ƽصҩá

ͪǽǿмأ޴ƼãͪۼúǿҲмػԣ ͪΪѡмأۼغʹƼãͪȻмƣ沪 лͬʱдƼءмغۼصáʴѡC 15⿼Ƥʼصʹ÷

ƤʼشƷжԸȾݿˣ˶ôҩʱ һ㲻3 գһƷڽ֯ۺ֧ Ĥסֶܰܰϸ԰Ѫȡ糿8 ʱһηãԡ 塢ƤƽᣬӦ١շҩɡϺãС ƷÿոҪʴѡB 20⿼ƤʼصĽ֤

ڸ߼ķƤʼؿƤʹܿ˸ѪѹӲˮ ס򲡻߽ãƤʼƹʵ׺ϳɣӸйƳԸƵ գԴ޸ڹۻ߽ãƤʼθθøķڣ谭֯޸ շθθ߽áܵ죬ż¾ʧշ

оʷáʴѡC 23⿼ȵصҩá

ȵضǴлӰҪǿǵתٽ֯ȡ ֽ⡢ԭĺϳɺ档ʴѡC 26⿼鵰ͬصҩ໤

ͬؿɽѪˮƽӦעѪǷӦķڼѪǣұƷ ӳѪգҩڼӦڼѪܣŮٰߣӦڼѪƼƣ ӦñƷʹתøAST ALTøøߣӦڼι ܡʴѡE

31⿼ҩIJӦ

ҩIJӦйӦӦϸȱ֢(ΪزӦҩ ʲȣӦͣҩӦ)״״ȣշ״ٹ ֢䱾Ϊ״ٹ֢ܿڿҩʴѡD 35⿼-øҩѪǵûơ

-øƼѪǵĻǣСƤˢ״Եྺˮˮ øӶˮ⼰ǵٶȲӻǵաʴѡD 37⿼鰬ĵע ƷҩӦʱΪ͵ѪǷտɿǼٻҩҩڼ Ż¡ظʹȼ֢״ӦעǷйԷӦ֢״ٲ ֻ߿ɲĿ壬ѪǿüӦѡҩƼ ĩڡ͸˻ʹñƷֲáƷƤע䡣 ѡE

41⿼״صҩ໤ ״ټصʳеĸơȽӵӰ죬Ӧڳոȫ ״ƣƳӦע⻼ĹܣĽʹʷĻӦôСʼд ܲȫٹܲȫĻ߻Լ״ƷӦ룬 ˣǰƤʼơĹܲȫļ֢״Ļߣ໤ҩ ڸŮڼ״ڼ䣬ܼ໤ɼ״ٹܹͻߣ ̥ɲӰ졣ʴѡC

52⿼࿹״ҩIJӦ Ӧ෢ҩʼ2 £ʮֳƤƤҩȡǴۺ Ƥסϸ١ϸ١ؽʹϸϸ ١ϸѪססټϸס ʴѡB

53⿼ҩ໤ ״ҩडͿϸ֢һ㷢ҩʼ ļ¡ϸȱַ֢ʽһͻȻһ㲻Ԥһ һаϸ٣ҩתϸȱ֢ҩڼ䣬Ӧÿ ܼ1 ΰϸҪʱƤʼơʴѡE 54⿼ٴӦá СҪƵԼ״ףҪƼ״صͷšʴѡC 55⿼鵰ͬصص㡣

ĵͬǽغͪܶͬãٽʵϳɡٽ ׳ٽʳٽ̼衢ٽϸʴѡA

56⿼͵⻯Ӧ֤

Ҫ(1)״Σ󣬵Ŀ״ÿǿúѸٸ֢״ ұͬʱӦҩ(2)״ٹ֢ܿǰ׼ʹ״֯ ӲѪ٣ڲгĽС״ٹ֢ܿǰȷһʱ ҩʹ֢״ͻлʻƺǰ2 ټõʴѡC 57⿼״ٹ֢ܿڿҩ ೣڼ״ٹ֢ܿڿƣ֢ͲԵߣС ԤԼ״ף״غ͵ɿڼ״ٹܵµ ʴѡD

58⿼ҩá

СǺϳɼ״ټصԭϣԤԼ״ףп״ã ҪƼ״ټصͷšʴѡE 59⿼ҩ໤

(1)ԿոѪǽϸѡóЧĸغ͸壻ͺѪѡöЧĸ ມͪ̽ϳҿոѪǽϸ߿ѡøб塢塢ء(2) ᡢжܲȫߣѡøͪͪΡ˫й򲡺 ܲȫʱӦȵơ(3)ԼļѪܼ Σߣѡ塢ຣѡб壻Լļߣڿʹ ȵأںѡҩ(4)б彵ǿʱ䳤һ ѪǣѡˣʹøбʱһҪעⲻɹֳֹ־õ ѪΣߡ(5)Ӧ״̬緢ȡԡȾʱڷҩ뻻 ơʴѡC

60⿼Ƽصҩá ƼشٽŮٵķͳ죬άŮԵڶмصЭͬʹӹĤ Ա仯γ¾ڡϴĴƼؿԴϵͳͨ GnRH ͷŶѣ֭ˮƽŴصйأƼ ˮãʹѪѹߡʴѡB 68⿼мصҩá

мܽӹƽصԣӹʹ̥ȫ ؿɴٽΪ׼мʹLH ڼ٣ѵ ãмؿɶԿȩͪٽйʴѡD 69⿼ҩûơ

ҩҪͨѣıӹҺʹӲ״͸ʹӹԭ 죬߲״ǸıӹѹܵĻʽ谭ܾѵ͡ʴѡ D

72⿼Ƽصص㡣

Ƽؾй㷺ҪãдٽάŮֳٺ͵ڶ ãڷڡѪܡлϵͳͳ켰ƤȸԵӰ졣 (1)ѳƼؿԴ̼ݷƼѪҺŨȵĸߵͿͨķʽٽ ƴټصͷţӶӰѳܡ(2)ѹܣƼܼѹ ٶȡ(3)ӹƼضӹĤƽĴлԴٽá(4)Ƽ ؿɴٽƤײϸֻԼǻܱ仯(5)٣ زԴ̼ٵܵҲܴٽݵķ֭ɡ(6) ƼдٽܵãʹպϺ͹ǻӰǵijӡڸ

ŮôƼƹ֢(7)ѪܣƼؿԽѪͨ͸ԣѪ嵨̴ ʴѡC

75⿼Ƽصҩ໤ ڴƼƿѪ˨˨¼ڿʼǰߵѪ˨¼ գȨףƼƿӹĤٰķգ˿ʼǰҲ ߸ĸգƼƿշѪֳѪҲ ڴڶҪų£ơʴѡA 76⿼мصҩá мάģ¾ںʹӹĤӹѪĤ Ϊֲܾ׼ֲܾʹ̥̣֮ӹ˷ԣ ʹ̥ȫƼعͬãʹ鷿ַΪ׼ʹӹ ڱպϣҺٱʹӲ״͸ʱͨԵĸãƴ ټصķڣáʴѡE

77⿼صǽѪҩٴӦص㡣 ˫ҩ֢2 򲡣ڷ߼ʳЧĻߡĿǰ Һ֯ƶָƼ˫Ϊغͷ2 򲡻߿ Ѫǵһҩມб͸ҪڵʳЧ2 ͶȵزܵĻߡʳ2 򲡡ʴѡD 81.⿼Ƽʹ÷

ʳ߲˺ˮйIJΣγɲԵĸΣʹƵ ٣ʳе֬γɶ۵ĸҲӰƵգӦעʳļ ʱ䡣峿˯ǰһΪѣԼʳԸյӰ죻ѡú Ƽ˯ǰá̼˥߽ѪʱӦڲзãǽ ѡA

83⿼֢ķࡣ

֢ɷΪ3 ࣺ(1)ԭԹ֢ں֢Թ ֢(2)̷Թ֢ijЩҩ糤ڴʹƤʼء Ӫȱ򲡡˥ߡԸβ״ٹܿ ۺĹɡ(3)طԹ֢ͳˣŴ ԼʷʴѡD

84⿼ǻҩá

ǻʳҩеĸڳбյĵڼͨ볦ϸڵİ ϣɴٽϸϳɸƽϵףӶٽϸĸתˣʹѪʴ ѡE

85⿼ƼIJӦ

øƼءʵȡż߸Ѫ֢жûҩ ָ߸Ѫ֢ΪηʳġŻ¡ءʹʧʴѡC 86⿼鰢ǻҩûơ

Ϊ(1)ССܶԸƵգƼ״ټ״ټغ ͷţƹա(2)ת-ºȵ-I ϳɣٽԭ ǻʵ׺ϳɡ(3)ڼƴлٽϸֻǿ񾭼Эԣ ٵ򡣹ʴѡD

87⿼άD IJӦ

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